Muscarinic Receptor

Cardiovascular effects of Sida cordifolia leaves extract in rats

Complementary and Alternative Medicine / Plant Biology / Electrocardiography / Blood Pressure / Animals / Male / Anesthesia / Heart rate / Malvaceae / Cardiovascular system / Plant extracts / Rats / Fitoterapia / Wistar Rats / Muscarinic Receptor / Plant Leaves / Bradycardia / Male / Anesthesia / Heart rate / Malvaceae / Cardiovascular system / Plant extracts / Rats / Fitoterapia / Wistar Rats / Muscarinic Receptor / Plant Leaves / Bradycardia

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Pharmacokinetics / In Vitro / Humans / Animals / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides / Drug Design / Acetylcholine / Bioavailability / Microdialysis / In Vivo / Rats / Rat / Cholinergic Receptor / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Chemical Synthesis / Area Under Curve / Benzamides

Benzylidene ketal derivatives as M2 muscarinic receptor antagonists

Organic Chemistry / Bioorganic and medicinal Chemistry / Muscarinic Receptor

The GABA uptake inhibitor β-alanine reduces pilocarpine-induced tremor and increases extracellular GABA in substantia nigra pars reticulata as measured by microdialysis

Neuroscience / Cognitive Science / Dialysis / Animals / Male / Acetylcholine / Substantia nigra / Tremor / High Performance Liquid Chromatography / High Pressure Liquid Chromatography / Microdialysis / Rats / Globus Pallidus / Pilocarpine / Motor Function / Basal ganglia / Neural pathways / Muscarinic Receptor / Statistical Methods for Neuroscience / Neurosciences / Parkinson Disease / Gamma-Aminobutyric Acid / Acetylcholine / Substantia nigra / Tremor / High Performance Liquid Chromatography / High Pressure Liquid Chromatography / Microdialysis / Rats / Globus Pallidus / Pilocarpine / Motor Function / Basal ganglia / Neural pathways / Muscarinic Receptor / Statistical Methods for Neuroscience / Neurosciences / Parkinson Disease / Gamma-Aminobutyric Acid

Benzylidene ketal derivatives as M2 muscarinic receptor antagonists

Organic Chemistry / Bioorganic and medicinal Chemistry / Muscarinic Receptor

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Humans / Animals / Drug Design / Acetylcholine / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides

3-(5-Alkylamino-4-isoxazolyl)-1,2,5,6-tetrahydropyridines: a novel class of central nicotinic receptor ligands

Organic Chemistry / Mass Spectrometry / Magnetic Resonance Spectroscopy / Cerebral Cortex / Animals / Male / Nicotinic Acetylcholine Receptors / Rats / Pyridines / Wistar Rats / Bioorganic and medicinal Chemistry / Muscarinic Receptor / Ligands / Male / Nicotinic Acetylcholine Receptors / Rats / Pyridines / Wistar Rats / Bioorganic and medicinal Chemistry / Muscarinic Receptor / Ligands

The GABA uptake inhibitor β-alanine reduces pilocarpine-induced tremor and increases extracellular GABA in substantia nigra pars reticulata as measured by microdialysis

Cognitive Science / Dialysis / Animals / Male / Substantia nigra / Tremor / High Pressure Liquid Chromatography / Microdialysis / Rats / Pilocarpine / Neural pathways / Muscarinic Receptor / Statistical Methods for Neuroscience / Neurosciences / Parkinson Disease / Gamma-Aminobutyric Acid / Tremor / High Pressure Liquid Chromatography / Microdialysis / Rats / Pilocarpine / Neural pathways / Muscarinic Receptor / Statistical Methods for Neuroscience / Neurosciences / Parkinson Disease / Gamma-Aminobutyric Acid

Muscarinic receptor subtype specificity of (N,N-dialkylamino)alkyl 2-cyclohexyl-2-phenylpropionates: cylexphenes (cyclohexyl-substituted aprophen analogs)

Organic Chemistry / Medicinal Chemistry / Pancreas / Animals / Male / Acetylcholine / Rats / Medicinal / Muscle contraction / Transfection / Muscarinic Receptor / Molecular Structure / Ileum / Acetylcholine / Rats / Medicinal / Muscle contraction / Transfection / Muscarinic Receptor / Molecular Structure / Ileum

Benzylidene ketal derivatives as M2 muscarinic receptor antagonists

Organic Chemistry / Bioorganic and medicinal Chemistry / Muscarinic Receptor

Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification

Organic Chemistry / Humans / Animals / Drug Design / Acetylcholine / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides / Microdialysis / Rats / Bioorganic and medicinal Chemistry / Structure activity Relationship / Muscarinic Receptor / Area Under Curve / Benzamides

Delayed Goblet Cell Hyperplasia, Acetylcholine Receptor Expression, and Worm Expulsion in SMC-Specific IL-4Rα–Deficient Mice

Microbiology / Immunology / Immune response / Medical Microbiology / Gene expression / Smooth muscle / Mice / Animals / Acetylcholine / Hyperplasia / Goblet Cells / Muscarinic Receptor / Smooth muscle / Mice / Animals / Acetylcholine / Hyperplasia / Goblet Cells / Muscarinic Receptor

Spontaneous Airway Hyperresponsiveness in Estrogen Receptor-α–deficient Mice

Electrophysiology / Cytokines / Inflammation / Sex Hormones / Estrogen Receptor / Serotonin / Lung Function / Mice / Female / Animals / American / Acetylcholine / Allergens / Lung / Estrogens / Trachea / Western blot / Peripheral nerves / Plethysmography / Muscarinic Receptor / Electric Field / Knockout Mice / Whole Body / bronchial hyperreactivity (BHR) / AIRWAY HYPERRESPONSIVENESS / Estrogen receptor alpha / Serotonin / Lung Function / Mice / Female / Animals / American / Acetylcholine / Allergens / Lung / Estrogens / Trachea / Western blot / Peripheral nerves / Plethysmography / Muscarinic Receptor / Electric Field / Knockout Mice / Whole Body / bronchial hyperreactivity (BHR) / AIRWAY HYPERRESPONSIVENESS / Estrogen receptor alpha

Delayed Goblet Cell Hyperplasia, Acetylcholine Receptor Expression, and Worm Expulsion in SMC-Specific IL-4Rα–Deficient Mice

Microbiology / Immunology / Immune response / Medical Microbiology / Gene expression / Smooth muscle / Mice / Animals / Acetylcholine / Hyperplasia / Goblet Cells / Muscarinic Receptor / Smooth muscle / Mice / Animals / Acetylcholine / Hyperplasia / Goblet Cells / Muscarinic Receptor

Spontaneous Airway Hyperresponsiveness in Estrogen Receptor-α–deficient Mice

Electrophysiology / Cytokines / Inflammation / Sex Hormones / Estrogen Receptor / Serotonin / Lung Function / Mice / Female / Animals / American / Acetylcholine / Allergens / Lung / Estrogens / Trachea / Western blot / Peripheral nerves / Plethysmography / Muscarinic Receptor / Electric Field / Knockout Mice / Whole Body / bronchial hyperreactivity (BHR) / AIRWAY HYPERRESPONSIVENESS / Estrogen receptor alpha / Serotonin / Lung Function / Mice / Female / Animals / American / Acetylcholine / Allergens / Lung / Estrogens / Trachea / Western blot / Peripheral nerves / Plethysmography / Muscarinic Receptor / Electric Field / Knockout Mice / Whole Body / bronchial hyperreactivity (BHR) / AIRWAY HYPERRESPONSIVENESS / Estrogen receptor alpha
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